2013 Publications

1)Yan He, Xinying Zhang, Nana Shen, Xuesen Fan*. Tunable synthesis of 3-acyl-2-naphthols and 3-substituted isocoumarins via Jones reagent promoted cascade reactions of 2-(4-hydroxy-but-1-ynyl) benzaldehydes.J. Org. Chem., 2013,78(20), 10178-10191.

2)Yan He, Xinying Zhang, Nana Shen, Xuesen Fan*. Synthesis of α-fluoroketones and α-fluoroenones in aqueous media.J. Flu. Chem.,2013,156(12), 9-14.

3)Yan He, Nana Shen, Xuesen Fan*, Xinying Zhang.Synthesis of β-fluoroenones and their reductive rearrangement in aqueous media.Tetrahedron,2013,69(41), 8818-8823.

4)Shenghai Guo*, Jiliang Wang, Xuesen Fan*, Xinying Zhang, Dongqiang Guo. Synthesis of pyrazolo [1,5-c]quinazoline derivatives through copper-catalyzed tandem reaction of 5-(2-bromoaryl)-1H- pyrazoles with carbonyl compounds and aqueous ammonia.J. Org. Chem.,2013,78(7), 3262-3270.

5)Qiang Wang, Zhouqing Xu, Xuesen Fan*. Selective synthesis of oxygen-containing heterocycles via tandem reactions of 1,2-allenic ketones with ethyl 4-chloroacetoacetate.RSC Adv.,2013,3(13), 4156- 4160.

6)Yan He, Xinying Zhang*, Liangyan Cui, Xuesen Fan*. Iodine-initiated domino reaction of hepta-1,2- dien-6-yn-4-ols and brønsted acid promoted cyclization of hepta-1,2,6-trien-4-ols leading to functionalized benzenes.Chem. Asian J.,2013,8(4), 717-722.

7)Xinying Zhang*, Xuefei Jia, Nan Liu, Xiaojie Guo, Yunping Song, Xuesen Fan*. 5-Hydroxypent-2-ene nitriles as precursors toward dihydropyranones, dienenitriles and functionalized naphthalenes.Tetrahedron,2013,69(26), 5374-5382.

8)Xinying Zhang*, Xiaojie Guo, Liangliang Fang, Yunping Song, Xuesen Fan*. Copper-catalyzed N- and O-arylation of amides: alternative approaches to 3,4-dihydroquinolin-2-ones, quinolin-2-ones, and 12H-chromeno[2,3-b]quinolin-12-ones.Eur. J. Org.Chem.,2013,(36), 8087-8093.

2012 Publications

1)Haiyun Xu, Xinying Zhang*, Yan He, Shenghai Guo, Xuesen Fan*. Tandem reaction of 3-hydroxyhexa -4,5-allenic esters: a novel access to diversely substituted 2H-pyran-2-ones and indenes.Chem. Commun., 2012,48(25), 3121-3123.

2)Yan He, Xinying Zhang*, Liangyan Cui, Jianji Wang, Xuesen Fan*. Catalyst-free synthesis of diversely substituted 6H-benzo[c]chromenes and 6H-benzo[c]chromen-6-ones in aqueous media under MWI.Green Chem., 2012,14(12), 3429-3435.

3)Xuesen Fan*, Yan He, Liangyan Cui, Shenghai Guo, Jianji Wang, Xinying Zhang*. Tandem reactions leading to benzo[c]chromen-6-ones and 3-substituted isocoumarins.Eur. J. Org. Chem., 2012 (4), 673-677.

4)Shenghai Guo*, Jiliang Wang, Dongqiang Guo, Xinying Zhang, Xuesen Fan*. Highly regioselective and practical synthesis of 1-acyl-5-hydroxypyrazolines and 1-acylpyrazoles from 1,2-allenic ketones and hydrazides.Tetrahedron, 2012,68(38), 7768-7774.

5)Shenghai Guo*, Jiliang Wang, Dongqiang Guo, Xinying Zhang, Xuesen Fan*. Synthesis of 3,5- disubstituted pyrazoles via cyclocondensation of 1,2-allenic ketones with hydrazines: application to the synthesis of 5-(5-methyl-pyrazol-3-yl)-2'-deoxycytidine.RSC Adv., 2012,2(9), 3772-3777.

2011 Publications

1)Xuesen Fan*, Yangyang Wang, Yingying Qu, Haiyun Xu, Yan He, Xinying Zhang*, Jianji Wang. Tandem reactions leading to bicyclic pyrimdine nucleosides and benzopyran-4-ones.J. Org. Chem., 2011,76(3), 982-985.

2)Xuesen Fan*, Yan He, Liangyan Cui, Xinying Zhang, Jianji Wang. Tandem reaction of 1,2-allenic ketone with α-halo ketone or α-halo ester in water: an efficient and sustainable synthesis of 1,3,4'-tricarbonyl compounds.Green Chem., 2011,13(11), 3218-3223.

3)Xinying Zhang*, Xuefei Jia, Liangliang Fang, Nan Liu, Jianji Wang, Xuesen Fan*. Tandem reactions of 1,2-allenic ketones leading to substituted benzenes and,-unsaturated nitriles.Org. Lett., 2011,13(19), 5024-5027.

4)Xinying Zhang*, Xuefei Jia, Jianji Wang, Xuesen Fan*. An economically and environmentally sustainable synthesis of 2-aminobenzothiazoles and 2-aminobenzoxazoles promoted by water.Green Chem., 2011,13(2), 413-418.

5)Xuesen Fan*, Xinying Zhang, Jianji Wang*. Recent progress in the green and efficient synthesis of biologically privileged scaffolds in ionic liquids.Curr. Org. Synth., 2011,8(5), 721-751.

6)Xinying Zhang*, Dongfang Li, Xuefei Jia, Jianji Wang, Xuesen Fan*. CuI/[bmim]OAc in [bmim]PF₆: a highly efficient and readily recyclable catalytic system for the synthesis of 2,3-disubstituted benzo[b] furans.Catal. Commun., 2011,12(9), 839-843.

7)Xuesen Fan*, Yan He, Xinying Zhang, Shenghai Guo. Synthesis of heteroaryl ketones via tandem reaction of 1,1-dibromoethenes.Tetrahedron, 2011,67(34), 6369-6374.

2010 Publications

1)XuesenFan*,Dong Feng, Yingying Qu, Xinying Zhang, Jianji Wang, Philippe M. Loiseau, Graciela Andrei,Robert Snoeck, Erik De Clercq.Practical and efficient synthesis of pyrano[3,2-c]pyridone,pyrano[4,3-b]pyran and their hybrids with nucleoside as potential antiviral and antileishmanial agents.Bioorg. Med. Chem. Lett.,2010,20(3), 809-813.

2)XuesenFan*,Yangyang Wang,Yan He, Xinying Zhang, Jianji Wang.Ru(III)-catalyzed oxidative reactionin ionic liquid: an efficient and practical route to 2-substituted benzothiazoles and their hybrids withpyrimidine nucleoside.Tetrahedron Lett.,2010,51(27), 3493-3496.

3)XuesenFan*,Yingying Qu, Yangyang Wang, Xinying Zhang, Jianji Wang.Ru(III)-catalyzed oxidation ofhomopropargyl alcohols in ionic liquid: an efficient and green route to 1,2-allenic ketones.TetrahedronLett.,2010,51(16), 2123-2126.

4)Xinying Zhang, Yingying Qu, XuesenFan*,C. Bores, Dong Feng, Graciela Andrei, Robert Snoeck, Erik DeClercq, Philippe M. Loiseau, Solvent-free synthesis of pyrimidine nucleoside-aminophosphonatehybrids and their biological activity evaluation.Nucleosides Nucleotides & Nucleic Acids,2010,29(8), 616-627.

5)张新迎,王洋洋,冯东,范学森*. 5-取代嘧啶核苷类似物的设计、合成及生物活性研究进展.有机化学, 2010, 30(6), 797-808.

6) XinyingZhang, Dongfang Li,Xuesen Fan*,XiaWang,XiaoyanLi,GuirongQu*,JianjiWang.Ionic liquidpromoted multi-component reaction: noveland efficient preparation of pyrazolo[3,4-b]pyridinone,pyrazolo[3,4-b]quinolinone and their hybrids with pyrimidinenucleoside.Mol. Diver.,2010, 14(1), 159-167.

2009 Publications

1) XinyingZhang,XiaoyanLi,DongfangLi,GuirongQu*,JianjiWang,PhillippeM.Loiseau,Xuesen Fan*.Ionic liquid mediated andpromoted eco-friendly preparation of thiazolidinone and pyrimidine nucleoside-thiazolidinone hybrids and their antiparasitic activities.Bioorg. Med.Chem.Lett.,2009, 19(22), 6280-6283.

2) XinyingZhang*,XiaoyanLi,Xuesen Fan*, Xia Wang, Jianji Wang, Guirong Qu,Controllable synthesis of pyrazolo[3,4-b]pyridines or substituted malononitrile derivatives through multi-component reactions in ionic liquid.Aust. J. Chem.,2009, 62(4), 382-388.

3)Xuesen Fan*, Dong Feng, Xia Wang, Yingying Qu, Xinying Zhang.Anovelpreparation ofpyridine–ureahybridsandelucidation oftheirstructures.Heteroatom Chem.,2009,20(6),362-368.

4) XinyingZhang*,XiaoyanLi,XuesenFan*,XiaWang,Dongfang,Li, Guirong Qu, Jianji Wang.Ionic liquid promoted preparation of 4H-thiopyran and pyrimidine nucleoside-thiopyran hybrids through one-pot multi-component reaction of thioamide.Mol. Diver.,2009, 13(1), 57-61.

2008 Publication

1)范学森*,张新迎,王霞,渠桂荣.碳环核苷的合成研究进展.有机化学, 2008, 28(11), 1888-1898.